Compile Data Set for Download or QSAR
maximum 50k data
Found 136 of ec50 data for complexid = 50008416
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222689(CHEMBL157774)
Affinity DataEC50: >30nMAssay Description:Agonistic activity towards vanilloid receptor, [Ca2+] influx in neonatal rat spinal sensory neuronal cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50222636(CHEMBL155978)
Affinity DataEC50: >30nMAssay Description:Agonistic activity towards vanilloid receptor, [Ca2+] influx in neonatal rat spinal sensory neuronal cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataEC50:  30nMAssay Description:In vitro agonist activity, increased [Ca2+] influx, at vanilloid receptor of rat dorsal root gangliaMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470963(CHEMBL146728)
Affinity DataEC50:  41nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470958(CHEMBL60744)
Affinity DataEC50:  56nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231166(CHEMBL58719)
Affinity DataEC50:  60nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231166(CHEMBL58719)
Affinity DataEC50:  60nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470962(CHEMBL144805)
Affinity DataEC50:  75nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231204(CHEMBL80662)
Affinity DataEC50:  100nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231186(CHEMBL309891)
Affinity DataEC50:  110nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470956(CHEMBL424317)
Affinity DataEC50:  130nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470976(CHEMBL146099)
Affinity DataEC50:  130nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231197(CHEMBL78616)
Affinity DataEC50:  160nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50055028(1-[4-(2-Amino-ethoxy)-3-methoxy-benzyl]-3-(4-tert-...)
Affinity DataEC50:  170nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20460((9Z)-N-[(4-hydroxy-3-methoxyphenyl)methyl]octadec-...)
Affinity DataEC50:  170nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20460((9Z)-N-[(4-hydroxy-3-methoxyphenyl)methyl]octadec-...)
Affinity DataEC50:  170nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231203(CHEMBL309532)
Affinity DataEC50:  180nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231198(CHEBI:46932 | Dihydrocapsaicin)
Affinity DataEC50:  190nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470955(CHEMBL147989)
Affinity DataEC50:  220nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231216(CHEMBL78895)
Affinity DataEC50:  240nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470957(CHEMBL147909)
Affinity DataEC50:  250nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231218(CHEMBL76848)
Affinity DataEC50:  270nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231175(CHEMBL76789)
Affinity DataEC50:  280nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231202(CHEMBL80404)
Affinity DataEC50:  290nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataEC50:  300nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50044753(2-(4-Hydroxy-3-methoxy-phenyl)-N-octyl-acetamide |...)
Affinity DataEC50:  300nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataEC50:  300nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataEC50:  300nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataEC50:  300nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470975(CHEMBL344133)
Affinity DataEC50:  320nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470967(CHEMBL147791)
Affinity DataEC50:  330nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231200(CHEMBL77292)
Affinity DataEC50:  350nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231155(CHEMBL77186)
Affinity DataEC50:  360nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231181(CHEMBL80637)
Affinity DataEC50:  360nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470968(CHEMBL356108)
Affinity DataEC50:  410nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470961(CHEMBL147716)
Affinity DataEC50:  480nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470969(CHEMBL357006)
Affinity DataEC50:  480nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50196351(1-(4-tert-Butyl-benzyl)-3-(4-hydroxy-3-methoxy-ben...)
Affinity DataEC50:  510nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231161(CHEMBL431379)
Affinity DataEC50:  530nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50044767(CHEMBL75124 | Hydroxymethoxybenzyl pelargonamide |...)
Affinity DataEC50:  550nMAssay Description:In vitro effective concentration for Ca++ uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50044767(CHEMBL75124 | Hydroxymethoxybenzyl pelargonamide |...)
Affinity DataEC50:  550nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231207(CHEMBL309275)
Affinity DataEC50:  620nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231213(CHEMBL310591)
Affinity DataEC50:  660nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231176(CHEMBL76476)
Affinity DataEC50:  670nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50470973(CHEMBL144093)
Affinity DataEC50:  710nMAssay Description:Compound tested in vitro for [Ca2+] influx into neonatal rat dorsal root ganglia (DRG)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231195(CHEMBL77089)
Affinity DataEC50:  1.08E+3nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231162(CHEMBL431788)
Affinity DataEC50:  1.16E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231153(CHEMBL312611)
Affinity DataEC50:  1.17E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231215(CHEMBL80341)
Affinity DataEC50:  1.24E+3nMAssay Description:In vitro effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in cultureMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1/2/4(Rattus norvegicus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50231169(CHEMBL76546)
Affinity DataEC50:  1.32E+3nMAssay Description:Effective concentration for [Ca2+] uptake into dorsal root ganglia neurones in rat cultured spinal sensory neuronesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 136 total ) | Next | Last >>
Jump to: